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L-152,804 is a potent, selective non-peptide neuropeptide Y Y5 receptor antagonist (Ki = 26 nM for hY5). Displays > 300-fold selectivity over hY1, hY2, and hY4 receptors. Causes weight loss in diet-induced obese mice by modulating food intake and energy expenditure. Centrally active upon oral administration in vivo.
| Molecular Weight | 366.46 |
| Formula | C23H26O4 |
| CAS Number | 6508-43-6 |
| Solubility (25°C) | DMSO 36.65 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Related Neuropeptide Receptor Products |
|---|
| JNJ-31020028
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22 rat); >100-fold selective versus human Y1/Y4/Y5 receptors. |
| BIBO 3304 trifluoroacetate
BIBO 3304 trifluoroacetate is a highly selective NPY Y 1 receptor antagonist. |
| CYM 9484
CYM 9484 is a potent NPY Y 2 receptor antagonist. |
| NTNCB hydrochloride
NTNCB hydrochloride is a potent and selective non-peptidic NPY Y 5 antagonist. |
| RF9
RF9 is a selective NPFF receptor antagonist (Ki values are 58 and 75 nM at hNPFF1 and hNPFF2 receptors respectively). |
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Products are for research use only. Not for human use. We do not sell to patients.
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