| Cat.No. | Name | Information |
|---|---|---|
| M50253 | Dimethindene maleate | Dimethindene maleate is a selective histamine H1 receptor antagonist with antihistamine activity.Dimethindene maleate may be used in studies related to allergic reactions. |
| M38976 | Diphenhydramine | Diphenhydramine is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine hydrochloride can across the ovine blood-brain barrier (BBB). |
| M30673 | Fexofenadine | Fexofenadine (MDL-16455) is an orally active and nonsedative H1 receptor antagonist. Fexofenadine can be used in allergic rhinitis and chronic idiopathic urticarial research. |
| M28480 | Clobenpropit dihydrobromide | Clobenpropit dihydrobromide is a potent histamine H3R antagonist/inverse agonist with a pEC50 of 8.07 for histamine H3LR. Clobenpropit dihydrobromide acts as partial agonist at histamine H4 receptors (Ki 13 nM). Clobenpropit dihydrobromide also binds to serotonin 5-HT3 receptors (Ki 7.4 nM) and α2A/α2C adrenoceptors (Ki 17.4/7.8 nM). Clobenpropit dihydrobromide increases apoptosis. |
| M22425 | Cetirizine | Cetirizine is a specific, orally active and long-acting histamine H1-receptor antagonist. Cetirizine marks antiallergic properties and inhibits eosinophil chemotaxis during the allergic response. |
| M22412 | Azelastine | Azelastine |
| M20516 | Ranitidine | Ranitidine is a histamine H2-receptor antagonist that inhibits stomach acid production. |
| M20511 | Betahistine | Betahistine is an orally active histamine H1 receptor agonist and a H3 receptor antagonist. |
| M13996 | Pitolisant hydrochloride | Pitolisant hydrochloride is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM). |
| M10773 | ABT-239 | ABT-239 is a novel, highly effective, non-imidazole H3R antagonist and antagonist of TRPV1. |
| M10717 | JNJ-5207852 | JNJ-5207852 IS HISTAMINE H3 RECEPTORS ARE SELECTIVELY EFFECTIVE ANTAGONISTS, WHICH ARE H AGAINST RATS AND HUMANS3 receptors pKi the values are 8.9 and 9.24, respectively. |
| M10715 | GSK189254A | GSK189254A (GSK189254) is a novel and highly effective selective H3 receptor antagonist for H3 in humans and ratshpi |
| M10714 | Pitolisant | Pitolisant is a potent and selective non-imidazole recombinant hentistamine H3 receptor reversed agonist,Ki 0.16 nM. |
| M10391 | Osthole | Osthole (Osthol) is a natural antihistamine alternative with potential inhibition of histamine H1 receptor activity. |
| M9459 | Mequitazine | Mequitazine is a potent, nonsedative and long-acting histamine H1 antagonist. |
| M9290 | S 38093 | S 38093 is an inverse agonist at histamine H3 receptors, displays a moderate affinity for rat, mouse and human H3 receptors with Ki of 8.8, 1.44 and 1.2µM, respectively. |
| M9172 | Emedastine Difumarate | Emedastine Difumarate is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. |
| M8821 | Triprolidine hydrochloride | Triprolidine hydrochloride is an orally active histamine H1 antagonist. Triprolidine hydrochloride has the function of spinal cord motor and sensory block. |
| M7895 | Levocetirizine dihydrochloride | Levocetirizine hydrochloride is a non-sedative antihistamine compound. |
| M6844 | JNJ 10191584 maleate | JNJ 10191584 maleate is a selective H 4 receptor antagonist; orally active. |
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