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Pitolisant hydrochloride is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
| Molecular Weight | 332.31 |
| CAS Number | 903576-44-3 |
| Solubility (25°C) | Water 90 mg/mL DMSO ≥ 43 mg/mL |
| Storage | 2-8°C, dry, sealed |
[3] Ulf Kallweit, et al. Pharmacological management of narcolepsy with and without cataplexy
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