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PF429242 dihydrochloride

Cat. No. M14435

All AbMole products are for research use only, cannot be used for human consumption.

PF429242 dihydrochloride Structure
Size Price Availability Quantity
1mg USD 40  USD40 In stock
5mg USD 95  USD95 In stock
10mg USD 135  USD135 In stock
25mg USD 285  USD285 In stock
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Quality Control & Documentation
Biological Activity

PF429242 dihydrochloride is a reversible and competitive SREBP site 1 protease (S1P) inhibitor with an IC50 of 175 nM.

Chemical Information
Molecular Weight 482.49
Formula C25H37Cl2N3O2
CAS Number 2248666-66-0
Form Solid
Solubility (25°C) DMSO ≥ 80 mg/mL
Water 50 mg/mL
Storage 2-8°C, dry, sealed
References

[1] Thais Tenorio Soares Fujii, et al. Microorganisms. Simvastatin Resistance of Leishmania amazonensis Induces Sterol Remodeling and Cross-Resistance to Sterol Pathway and Serine Protease Inhibitors

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Keywords: PF429242 dihydrochloride supplier, FAS, inhibitors, activators

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