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MK 0893 is a potent and selective glucagon receptor antagonist with an IC50 of 6.6 nM.
| Molecular Weight | 588.48 |
| CAS Number | 870823-12-4 |
| Solubility (25°C) | DMSO ≥ 33.33 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] Ali Jazayeri, et al. Extra-helical binding site of a glucagon receptor antagonist
[3] Hong-Ping Guan, et al. Glucagon receptor antagonism induces increased cholesterol absorption
[4] Songnian Lin, et al. A novel series of indazole-/indole-based glucagon receptor antagonists
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