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M435-1279 

Cat. No. M31238

All AbMole products are for research use only, cannot be used for human consumption.

M435-1279  Structure
Size Price Availability Quantity
5mg USD 140  USD140 In stock
10mg USD 220  USD220 In stock
25mg USD 420  USD420 In stock
50mg USD 700  USD700 In stock
100mg USD 1100  USD1100 In stock
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Quality Control & Documentation
Biological Activity

M435-1279 is a UBE2T inhibitor. M435-1279 inhibits the Wnt/β-catenin signaling pathway hyperactivation through blocking UBE2T-mediated degradation of RACK1.

Chemical Information
Molecular Weight 419.47
Formula C18H17N3O5S2
CAS Number 1359431-16-5
Form Solid
Solubility (25°C) DMSO 50 mg/mL (Need ultrasonic)
Storage 4°C, protect from light
References

[1] Yang Wang, et al. Drug Des Devel Ther. UBE2T Promotes Temozolomide Resistance of Glioblastoma Through Regulating the Wnt/β-Catenin Signaling Pathway

[2] Shusheng Cai, et al. Dis Markers. Transcription Activation of Rab8A by PEA3 Augments Progression of Esophagus Cancer by Activating the Wnt/ β-Catenin Signaling Pathway

[3] Zeyuan Yu, et al. Oncogene. A novel UBE2T inhibitor suppresses Wnt/β-catenin signaling hyperactivation and gastric cancer progression by blocking RACK1 ubiquitination

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  Catalog
Abmole Inhibitor Catalog




Keywords: M435-1279  supplier, E1/E2/E3 Enzyme, inhibitors, activators

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