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Drinabant

Cat. No. M29983

All AbMole products are for research use only, cannot be used for human consumption.

Drinabant Structure
Synonym:

AVE1625

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Quality Control & Documentation
Biological Activity

Drinabant (AVE1625) is an orally active CB1 receptor antagonist. Drinabant (AVE1625) inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R.

Chemical Information
Molecular Weight 497.38
Formula C23H20Cl2F2N2O2S
CAS Number 358970-97-5
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Phil Skolnick, et al. J Neural Transm (Vienna). Cannabinoid1 (CB-1) receptor antagonists: a molecular approach to treating acute cannabinoid overdose

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Keywords: Drinabant, AVE1625 supplier, Cannabinoid, inhibitors, activators

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