Free shipping on all orders over $ 500

AM251

Cat. No. M2379

All AbMole products are for research use only, cannot be used for human consumption.

AM251 Structure
Size Price Availability Quantity
5mg USD 50  USD50 In stock
10mg USD 85  USD85 In stock
50mg USD 290  USD290 In stock
100mg USD 480  USD480 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

AM251 block the inhibitory effects of endocannabinoids and synthetic cannabinoid agonists on transmitter release through an action at presynaptic cannabinoid 1 receptors in brain.

Chemical Information
Molecular Weight 555.24
Formula C22H21Cl2IN4O
CAS Number 183232-66-8
Solubility (25°C) DMSO 30 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Ins B Correia-S, et al. AM251, a cannabinoid receptor 1 antagonist, prevents human fibroblasts differentiation and collagen deposition induced by TGF-β - An in vitro study

[2] Inmaculada Ruz-Maldonado, et al. The cannabinoid ligands SR141716A and AM251 enhance human and mouse islet function via GPR55-independent signalling

[3] Tomoyo Yoshinaga, et al. AM251 Suppresses Epithelial-Mesenchymal Transition of Renal Tubular Epithelial Cells

[4] Sara Carpi, et al. AM251 induces apoptosis and G2/M cell cycle arrest in A375 human melanoma cells

[5] Izabela Bialuk, et al. AM251, cannabinoids receptors ligand, improves recognition memory in rats

Related Cannabinoid Products
Org 27569

Org 27569 is a potent and selective allosteric modulator of the cannabinoid CB1 receptor.

AM1241

AM1241 is a cannabinoid CB2 receptor selective agonist.

CP 945598 hydrochloride

CP 945598 hydrochloride is a selective and high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively).

AM-2201

AM-2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively.

BML-190

BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.

  Catalog
Abmole Inhibitor Catalog




Keywords: AM251 supplier, Cannabinoid, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.