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BI8622 is a specific inhibitor of the ubiquitin ligase HUWE1 with an IC50 of 3.1 μM.
| Molecular Weight | 426.51 |
| CAS Number | 1875036-74-0 |
| Solubility (25°C) | DMSO 90 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Jing Zhang, et al. Retinitis pigmentosa 2 pathogenic mutants degrade through BAG6/HUWE1 complex
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