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Adomeglivant

Cat. No. M13966

All AbMole products are for research use only, cannot be used for human consumption.

Adomeglivant Structure
Synonym:

LY2409021

Size Price Availability
5mg USD 90  USD90 4-7 Days
10mg USD 150  USD150 4-7 Days
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Quality Control & Documentation
Biological Activity

Adomeglivant (LY2409021) is a potent, selective glucagon receptor (GluR) allosteric antagonist. Adomeglivant is widely used in the research for type 2 diabetes mellitus.

Chemical Information
Molecular Weight 555.63
CAS Number 1488363-78-5
Solubility (25°C) DMSO ≥ 90 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Sofie Hdersdal, et al. The glucagon receptor antagonist LY2409021 has no effect on postprandial glucose in type 2 diabetes

[2] Sofie Hdersdal, et al. The Role of Glucagon in the Acute Therapeutic Effects of SGLT2 Inhibition

[3] Wyatt J Roth, et al. A Demonstration of Mixing Robustness in a Direct Compression Continuous Manufacturing Process

[4] Yong Li, et al. Efficient Synthesis of β-CF3/SCF3-Substituted Carbonyls via Copper-Catalyzed Electrophilic Ring-Opening Cross-Coupling of Cyclopropanols

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Keywords: Adomeglivant, LY2409021 supplier, Glucagon Receptor, inhibitors, activators

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