All AbMole products are for research use only, cannot be used for human consumption.
Vapreotide acetate (BMY-41606 acetate; RC160 acetate) is a neurokinin-1 (NK1) receptor antagonist with IC50 value of 330 nM. Vapreotide inhibits SP-induced IL-8 and MCP-1 production in HEK293-NK1R and U373MG cell lines. Vapreotide also inhibits HIV-1 infection of human MDM in vitro, an effect that is reversible by SP pretreatment. Vapreotide inhibits serum-induced proliferation of CHO cells expressing SSTR2 and SSTR5 with EC50 of 53 and 150 pM, respectively.
| Molecular Weight | 1191.39 |
| Formula | C59H74N12O11S2 |
| CAS Number | 849479-74-9 |
| Solubility (25°C) | Water 11 mg/mL |
| Storage | -20°C, sealed |
| Related Neurokinin Receptor Products |
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| Monohydroxy Netupitant
Monohydroxy Netupitant is the metabolite of Netupitant, which is a highly selective NK1 receptor antagonist. |
| Aprepitant
Aprepitant (Emend) is an antiemetic chemical compound that belongs to a class of compounds called substance P antagonists (SPA). |
| Maropitant
Maropitant (Cerenia) is a novel, selective neurokinin type-1 (NK1) receptor antagonist. |
| Eprazinone dihydrochloride
Eprazinone is a mucolytic. |
| Fosaprepitant dimeglumine salt
Fosaprepitant is a water-soluble phosphoryl procompound for Aprepitant which is a NK1 antagonist.*The compound is unstable in solutions, freshly prepared is recommended |
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Products are for research use only. Not for human use. We do not sell to patients.
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