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Thiethylperazine 

Cat. No. M28383

All AbMole products are for research use only, cannot be used for human consumption.

Thiethylperazine  Structure
Size Price Availability Quantity
5mg USD 95  USD95 In stock
10mg USD 145  USD145 In stock
25mg USD 280  USD280 In stock
50mg USD 430  USD430 In stock
100mg USD 650  USD650 In stock
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Quality Control & Documentation
Biological Activity

Thiethylperazine, a phenothiazine derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist. Thiethylperazine is also a selective ABCC1activator that reduces amyloid-β (Aβ) load in mice. Thiethylperazine has anti-emetic, antipsychotic and antimicrobial effects.

Chemical Information
Molecular Weight 399.62
Formula C22H29N3S2
CAS Number 1420-55-9
Form Solid
Solubility (25°C) DMSO 100 mg/mL (ultrasonic)
Storage 4°C, protect from light
References

[1] Michael Wölfl-Duchek, et al. Int J Mol Sci. Use of PET Imaging to Assess the Efficacy of Thiethylperazine to Stimulate Cerebral MRP1 Transport Activity in Wild-Type and APP/PS1-21 Mice

[2] No authors listed. Thiethylperazine

[3] A E Czeizel, et al. BJOG. Case-control study of teratogenic potential of thiethylperazine, an anti-emetic drug

[4] R Sulkava. Acta Neurol Scand. Thiethylperazine and tardive dyskinesia

[5] B Larkman. Can J Psychiatr Nurs. Thiethylperazine--Torecan

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Keywords: Thiethylperazine  supplier, Dopamine Receptor, inhibitors, activators

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