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Terlakiren

Cat. No. M42603

All AbMole products are for research use only, cannot be used for human consumption.

Terlakiren Structure

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Quality Control & Documentation

COA
MSDS

Product Information

Biological Activity

Terlakiren (CP-80,794) is an orally active inhibitor of renin.

Chemical Information

Molecular Weight	620.8
Formula	C31H48N4O7S
CAS Number	119625-78-4
Storage	Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month

References

[1] Serdar Durdagi et al. Mol Inform. Screening of Clinically Approved and Investigation Drugs as Potential Inhibitors of SARS-CoV-2: A Combined in silico and in vitro Study

[2] M L Mangiapane et al. Clin Exp Hypertens. Role of nitric oxide in responses to renin-angiotensin system inhibition in sodium-depleted guinea pig and rat

[3] R P Shannon et al. Cardiovasc Res. Effects of renin inhibition compared to angiotensin converting enzyme inhibition in conscious dogs with pacing-induced heart failure

[4] D J Hoover et al. Adv Exp Med Biol. Discovery of inhibitors of human renin with high oral bioavailability

[5] A A Fossa et al. J Cardiovasc Pharmacol. Synergistic effect on reduction in blood pressure with coadministration of the renin inhibitor, CP-80,794, and the angiotensin converting enzyme inhibitor, captopril

Related Renin Products
Aliskiren Hemifumarate Aliskiren hemifumarate is a direct renin inhibitor with IC50 of 1.5 nM.
Aliskiren Aliskiren(CGP 60536) is a direct renin inhibitor with IC50 of 1.5 nM.
Renin substrate 1 Renin substrate 1 is a renin substrate with high affinity to the enzyme.

Catalog

Abmole Inhibitor Catalog

Keywords: Terlakiren supplier, Renin, inhibitors, activators

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