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TC LPA5 4 is a specific non-lipid LPA5 (GPR92) antagonist (IC50=0.8 μM in LPA5-RH7777 cells). Shows selectivity for LPA5 against 80 other screening targets.TC LPA5 4 was shown to inhibit LPA-induced aggregation of isolated human platelets.TC LPA5 4 inhibits proliferation and migration of thyroid cancer cells.
| Molecular Weight | 410.89 |
| Formula | C23H23ClN2O3 |
| CAS Number | 1393814-38-4 |
| Solubility (25°C) | DMSO ≥ 60 mg/mL |
| Storage | 2-8℃, protect from light, dry, sealed |
| Related LPL Receptor Products |
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| Ki16425
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| Ki16198
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| GSK-2018682
This compound belongs to the class of organic compounds known as n-alkylindoles. These are compounds containing an indole moiety that carries an alkyl chain at the 1-position. |
| H2L5186303
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| AM095 sodium
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