Free shipping on all orders over $ 500

Proglumide sodium salt

Cat. No. M7161

All AbMole products are for research use only, cannot be used for human consumption.

Proglumide sodium salt Structure
Size Price Availability Quantity
10mg USD 25  USD25 In stock
25mg USD 55  USD55 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Proglumide sodium salt is a non-selective, orally active cholecystokinin (CCK) antagonist. Proglumide sodium inhibits CCK-stimulated amylase secretion and prevents CCK-induced 2-deoxyglucose uptake in mouse pancreatic acini. Proglumide sodium blocks growth of HT29 colon carcinoma cells in response to gastrin 17 treatment.

Chemical Information
Molecular Weight 356.39
Formula C18H25N2NaO4
CAS Number 99247-33-3
Solubility (25°C) Water 35.64 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Qiao, et al. Med Chem. Triphenylethanamine derivatives as cholesteryl ester transfer protein inhibitors: discovery of N-[(1R)-1-(3-cyclopropoxy-4-fluorophenyl)-1-[3-fluoro-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-2-phenylethyl]-4-fluoro-3-(trifluoromethyl)benzamid J.

Related Cholecystokinin Receptor Products
Pentagastrin

Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally.

Lintitript

Lintitript (SR 27897) is a highly potent, selective, orally active, competitive and non-peptide cholecystokinin (CCK1) receptor antagonist with an EC50 of 6 nM and a Ki of 0.2 nM. Lintitript displays > 33-fold selectivity more selective for CCK1 than CCK2 receptors (EC50 value of 200 nM).

Lorglumide sodium salt

Lorglumide (CR-1409) sodium salt is a potent cholecystokinin (CCK) receptor antagonist.

Gastrin-I (human)

Gastrin-I (human) is the endogenous peptide produced in the stomach, which increases gastric acid secretion via cholecystokinin 2 (CCK2) receptor.

Gastrin I (rat) TFA

Gastrin I (rat) TFA is a peptide hormone, which can stimulate gastric acid secretion potently.

  Catalog
Abmole Inhibitor Catalog




Keywords: Proglumide sodium salt supplier, Cholecystokinin Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.