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PF-9363

Cat. No. M40815

All AbMole products are for research use only, cannot be used for human consumption.

PF-9363 Structure
Synonym:

CTx-648

Size Price Availability Quantity
1mg USD 80  USD80 In stock
5mg USD 200  USD200 In stock
10mg USD 300  USD300 In stock
50mg USD 650  USD650 In stock
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Quality Control & Documentation
Biological Activity

PF-9363 is a first-in-class, orally active, highly selective KAT6A/B inhibitor for studies related to ER-positive breast cancer.

Chemical Information
Molecular Weight 444.46
Formula C20H20N4O6S
CAS Number 2569009-58-9
Form Solid
Solubility (25°C) DMSO 50 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Shikhar Sharma et al. Cell Chem Biol. Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer

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Keywords: PF-9363, CTx-648 supplier, Histone Acetyltransferase, inhibitors, activators

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