All AbMole products are for research use only, cannot be used for human consumption.
For this product's availability, delivery time and price, please email [email protected] directly or click the "Inquiry Now" button below.
PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; PD176252 is also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells.
| Molecular Weight | 584.67 |
| Formula | C32H36N6O5 |
| CAS Number | 204067-01-6 |
| Form | Solid |
| Solubility (25°C) | DMSO 115 mg/mL (ultrasonic) |
| Storage | 4°C, sealed |
| Related Bombesin Receptor Products |
|---|
| MK-5046
MK-5046 is an orally active, potent, selective agonist of the orphan G protein-coupled receptor bombesin receptor subtype-3 (BRS-3) that is under evaluation for treatment of obesity. |
| Kuwanone H
Kuwanone H |
| ML-18
ML18 is Bombesin receptor subtype 3 (BRS-3) antagonist (IC50 = 4.8 μM). |
| Bombesin
Bombesin is a tetradecapeptide, which plays an important role in the release of gastrin and the activation of G-protein receptors. |
| Ranatensin
Ranatensin is a undecapeptide and a Bombesin Receptor angonist, which could maintain the dynamic balance of animal blood pressure, without cross-tachyphylaxis with Angiotensin amide, Bradykinin, or Norepinephrine. |
All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.
