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Ocedurenone

Cat. No. M40521

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Ocedurenone Structure
Synonym:

KBP-5074

Price and Availability

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Quality Control & Documentation
Biological Activity

Ocedurenone is a novel nonsteroidal salicorticoid receptor (MR) antagonist that may be used in studies related to kidney disease.

Chemical Information
Molecular Weight 504.02
Formula C28H30ClN5O2
CAS Number 1359969-24-6
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Duygu Koca et al. Steroids. Molecular pharmacology of mineralocorticoid receptor antagonists: The role of co-regulators

[2] George L Bakris et al. Am J Hypertens. Efficacy and Safety of Ocedurenone: Subgroup Analysis of the BLOCK-CKD Study

[3] Ping Wang et al. Eur J Drug Metab Pharmacokinet. Pharmacokinetics and Drug-Drug Interaction of Ocedurenone (KBP-5074) in vitro and in vivo

[4] Panagiotis I Georgianos et al. Nephrol Dial Transplant. Hypertension in chronic kidney disease - treatment standard 2023

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Keywords: Ocedurenone, KBP-5074 supplier, Mineralocorticoid Receptor, inhibitors, activators

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