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LBW242, a 3-mer and Smac mimetic, is a potent and orally active proapoptotic IAP inhibitor. LBW242 shows effects on mutant FLT3-expressing cells. LBW242 has activity against multiple myeloma, and potentiates TRAIL- and anticancer agent-mediated cell death of ovarian cancer cells.
| Molecular Weight | 454.65 |
| Formula | C27H42N4O2 |
| CAS Number | 867324-12-7 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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