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GSK2239633A is a CC-chemokine receptor 4 (CCR4) antagonist, which inhibits the binding of [125I]-TARC to human CCR4 with a pIC50 of 7.96 ± 0.11.
| Molecular Weight | 549.06 |
| Formula | C24H25ClN4O5S2 |
| CAS Number | 1240516-71-5 |
| Form | Solid |
| Solubility (25°C) | DMSO ≥ 250 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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