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DAPTA is a water soluble potent, selective CCR5 inhibitor which potently inhibits specific CD4-dependent binding of gp120 Bal (IC50 = 0.06 nM) and CM235 (IC50 = 0.32 nM) to CCR5.
| Molecular Weight | 856.88 |
| Formula | C35H56N10O15 |
| CAS Number | 106362-34-9 |
| Solubility (25°C) | Water 50 mg/mL |
| Storage | Store at ≤ -20°C, dry, sealed |
| Related CCR Products |
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| INCB3284 dimesylate
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