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Chiglitazar

Cat. No. M30564

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Chiglitazar Structure
Synonym:

Carfloglitazar

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Quality Control & Documentation
Biological Activity

Chiglitazar (Carfloglitazar) is a PPARα/γ dual agonist, with EC50s of 1.2, 0.08, 1.7 μM for PPARα, PPARγ and PPARδ, respectively.

Chemical Information
Molecular Weight 572.62
Formula C36H29FN2O4
CAS Number 743438-45-1
Form Solid
Solubility (25°C) DMSO 100 mg/mL (ultrasonic)
Storage 4°C, protect from light, dry, sealed
References

[1] Ralph A DeFronzo. Sci Bull (Beijing). Chiglitazar: a novel pan-PPAR agonist

[2] Emma D Deeks. Drugs. Chiglitazar: First Approval

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  Catalog
Abmole Inhibitor Catalog




Keywords: Chiglitazar, Carfloglitazar supplier, PPAR, inhibitors, activators

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