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BMS-986235

Cat. No. M21272

All AbMole products are for research use only, cannot be used for human consumption.

BMS-986235 Structure
Synonym:

LAR-1219

Price and Availability

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Quality Control & Documentation
Biological Activity

BMS-986235/LAR-1219 is an FPR1-sparing FPR2-selective agonist designed to help address chronic inflammation/promote wound healing to prevent serious complications such as heart failure.

Chemical Information
Molecular Weight 361.34
Formula C18H17F2N3O3
CAS Number 2253947-47-4
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Ricardo A Garca, et al. JACC Basic Transl Sci. Selective FPR2 Agonism Promotes a Proresolution Macrophage Phenotype and Improves Cardiac Structure-Function Post Myocardial Infarction

[2] John Lupisella, et al. ACS Pharmacol Transl Sci. Molecular Mechanisms of Desensitization Underlying the Differential Effects of Formyl Peptide Receptor 2 Agonists on Cardiac Structure-Function Post Myocardial Infarction

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  Catalog
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Keywords: BMS-986235, LAR-1219 supplier, FPR, inhibitors, activators

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