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ACH-000143 

Cat. No. M29376

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ACH-000143  Structure

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Quality Control & Documentation
Biological Activity

ACH-000143 is a potent and orally active melatonin receptor agonist, with EC50 values of 0.06 nM and 0.32 nM for MT1 and MT2, respectively.

Chemical Information
Molecular Weight 297.74
Formula C13H16ClN3O3
CAS Number 2225836-30-4
Form Solid
Solubility (25°C) DMSO 50 mg/mL (ultrasonic)
Storage 4°C, protect from light
References

[1] Marcos Antonio Ferreira Jr, et al. J Med Chem. Discovery of ACH-000143: A Novel Potent and Peripherally Preferred Melatonin Receptor Agonist that Reduces Liver Triglycerides and Steatosis in Diet-Induced Obese Rats

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  Catalog
Abmole Inhibitor Catalog




Keywords: ACH-000143  supplier, Melatonin Receptor, inhibitors, activators

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